Phenibut Uses and Benefits
People will always search for a magic capsule that will make them smarter, concentrated, attentive, and able to manage any scope of work. Now it seems to be true that a new wave of interest arose around Phenibut, a brain boosting substance synthesized in the last century.
In the myriad of lab-developed medicines, Phenibut really possesses the properties of a “smart drug.”
If you have never heard of this outstanding substance, it high time to take a deeper look at its benefits. Who knows, maybe it can turn someone’s life upside down?
What Is Phenibut?
Phenibut is a chemical derived from gamma-Aminobutyric acid (GABA). GABA is a neurotransmitter which decreases anxiety and naturally controls the neuronal excitability of the central nervous system (CNS). In other words, it ensures that the human brain does not become hyperactive. Phenibut is commercially available under the names of Fenibut, Noofen, and Anvifen.
GABA supplements cross the blood-brain barrier less efficiently as Phenibut, and sometimes they are used together in a stack.
Phenibut supplementation greatly affects CNS activity and performs two main functions:
- as a powerful anxiolytic, it is used to cure neuroses, insomnia, irritability, hyperactivity, panic attacks, and various stress disorders;
- as a strong nootropic, it improves attention, motivation, memory, and concentration.
Most such compounds impair human brain functions, but Phenibut is different and doesn’t negatively affect cognitive abilities. Users get more control over their stress level, which usually leads to sleep deprivation and anxiety. Phenibut improves sleep patterns and promotes a better sleep quality, so its users wake up rested.
This drug also prevents neuronal cells’ damage, which happens each time our stress level is high. Due to an increased dopamine level, people get a more positive mood and subsequent higher motivation.
Phenibut sedative’s impact can be compared to that of alcohol, but without the depressant side effects. This drug provides better focus and a calm effect, as well as increases sociability without negative reactions produced by ethanol and caffeine. It is ideal for people who feel socially nervous and anxious, so they get a better control over their thoughts and feelings. Phenibut is a great help for self-conscious people inclined to overthink.
Phenibut was first discovered and synthesized in 1963 in St. Petersburg, Russia, by Professor V.V. Perekalin at the Herzen State Pedagogical University of Russia. This experimental medicine with tranquilizing effects (in early publications called phenigamma) was developed for young patients under psychiatric therapy.
Only in 1975 did this drug became known as Phenibut and was widely used to cure emotional and mental malfunctions.
Unlike regular anti-anxiety drugs, which cause drowsiness, this medicine produced no negative effects on performance level. It was effective to cope with fear, insomnia, stress, tension, and it even recorded numerous reports of increased cognition.
Phenibut was taken by Russian astronauts to combat insomnia and anxiety. It became an essential thing in medical kits on Russian space flights. It is still being used as psychotropic medicine sold under prescription. It is currently known as a sleep aid, mood enhancer, and recovery booster. Due to its memory recall benefits, Phenibut attracts numerous customers to the “smart drug” market.
How Does This Nootropic Work?
Phenibut is similar in its structure to the neurotransmitter γ-aminobutyric acid (or GABA), which is important for decreasing anxiety and excitability. GABA is manufactured in the human body and is not very effective in crossing the blood-brain barrier, but Phenibut is more successful at it.
The blood-brain barrier is a significant mechanism of the human body which prevents harmful elements and toxins travelling through the blood from reaching the brain. Phenibut can easily enter the brain through a phenyl ring and eliminate social inhibition and anxiety. Along with GABA, it naturally balances the effects of different elements, which trigger neurons. When neurons become overstimulated, it causes the feelings of restlessness and worry. Phenibut is successful in restoring this balance.
The drug is able to stimulate dopamine receptors responsible for mood elevation. Due to an increased dopamine level, users experience a positive mood and a higher motivation level.
As a synthetic GABA form, it is not selective and stimulates both GABA-A and GABA-B receptors. It also results in the feelings of relaxation and calmness.
Its beneficial effects are not properly studied in human trials and need further investigation. Phenibut is used as a psychotropic medicine, which means it can alter user’s mental state. It does help patients in overcoming unpleasant mental disease symptoms. Still, it lacks academically published reports and profound information to be used on a therapeutic basis for human beings.
How to Take Phenibut?
Phenibut is usually taken orally, because other administration forms can be rather dangerous. With Phenibut injections, users may acquire vascular damage.
As this powder is a water-soluble substance, some people find it more convenient to buy Phenibut in bulk and dissolve it into water. It is better to consume it with light food, because heavy meals may slow down tablet absorption.
Phenibut has a rather high pH level, which creates its bitter taste. Most consumers still prefer to buy the powder in capsules.
The drug takes longer for the effects to come out, sometimes up to 4 hours. If users divide a daily Phenibut intake dose into several doses, the next portion should be taken 4 hours after the previous.
The half-life of Phenibut is 5-6 hours, but its residual effects are reported within the next 24 hours.
Do not mix Phenibut with other similar substances, as it may provoke respiratory depression. Alcohol may do the same, as it increases user’s chances to become unconscious. This drug interacts with other tablets, and it causes negative reactions for some diseases, for example, it cannot be used by Parkinson’s sufferers. Phenibut can cause overdosing symptoms if combined with other CNS depressants (as opioids) or sedatives.
An appropriate daily dose of Phenibut depends on different factors that include the user’s health, age, gender, and health conditions. It is important to speak to a doctor before the first use and follow all his recommendations on how to take it. That is an important warning, because abuse may lead to drug dependence.
An average advised dosage is 250 mg, but lower doses are highly welcomed to start. A proper dose can be calculated as 15-17 mg per pound of body weight. A healthy man in his late teens can take 250 mg, which are subdivided into 3 doses during one day.
Female patients are recommended lower doses, calculated as 8-10 mg per pound of body weight. Anyway, it is not a standard and depends on each woman’s health. A healthy woman may take 100 mg as a daily dose subdivided into 3 portions.
Phenibut dosage also depends on the concern or disease that is being treated. To cure anxiety and stress, take lower doses to avoid drowsiness. Insomnia patients are prescribed higher doses. Again, an excessive serving can create a hyperarousal state and the inability to fall asleep. At the same time, people who usually don’t suffer from stress disorders may feel no effect unless they consume a high dose.
Most studies recommend using no more than 300 mg of Phenibut a day as a safe dose, which induces no psychological adverse effects. However, further research indicates that consumed 10 days in a row, this portion is likely to cause addiction. Therefore, the best way is to underdose to avoid side effects.
In order avoid developing a tolerance to the drug, some users take it for 2 weeks and pause for the next 2 weeks.
Remember that Phenibut is a drug and cannot be used as a daily supplement. Take it only when it is really required.
If Phenibut is consumed as recommended by doctors, it is safe for users. If the maximum dose is exceeded, the following symptoms are likely to occur:
- loss of balance;
- memory loss;
Long-term usage may cause dependence because of increased tolerance of the body to the substance. If patients stop using Phenibut abruptly, they may acquire withdrawal symptoms:
- muscle spasms;
- panic attacks;
- vivid dreams;
In this case, quit using the drug for a few days to diminish tolerance to the medicine. By the following intake, patients can feel limb pain or numbness after sleep. These withdrawal effects will disappear after a dose reduction.
Rare adverse reactions include lethargy, blood pressure decrease, shallow irregular breathing, and increased sweating.
These reported symptoms uncover the truth of the unregulated internet drug market that ensures no quality standards. Buy Phenibut only from trusted suppliers.
Are There Any Other Effective Brain Boosters?
The modern pharmacological market is overburdened with various supplements and drugs that are introduced to us as cognitive boosters. Before we fuel our brain with some risky substances that are labeled as brain enhancers, let us analyze what particular elements nourish our brain cells. Most ingredients have proven scientific evidence and are considered safe to combat memory problems.
The basic action mechanism of almost all famous supplements is that they work on the neuron level by inhibiting or increasing the production of particular enzymes in the brain. The correct balancing of an amount of these enzymes helps to regulate our mental activity.
Some of the elements given below are the most prominent, which are worth mentioning:
- dimethylaminoethanol or DMAE (This amino acid provides sound brain cell operation and stimulates oxygen supply to the brain.);
- docosahexaenoic acid or DHA (This omega-3 fatty acid takes part in the formation of new brain cells. It is helpful for dementia and depression.);
- acetyl-L-carnitine or ALC (This amino acid diminishes brain cell damage and improves alertness and learning abilities.);
- citicoline (This element protects the brain from free radical damage and aging and treats memory loss.);
- tryptophan (By increasing serotonin levels, this amino acid improves sleep processes, mood, short-term, and long-term memory.);
- phosphatidylserine or PS (This phospholipid reduces stress hormones and keeps toxins out of the brain.);
- choline (This nutrient helps in brain development and proper brain cell functioning.);
- L-theanine (By enhancing dopamine and serotonin levels, this amino acid sharpens our focus, as well as promotes motivation and attention.);
- alpha-glycerophosphocholine (This supplement copes with mental decline and restores the brain after heart attacks.)
Talk to a physician and work out your individual brain supplementation scheme regarding your needs and demands.
Herbs, Vitamins and Minerals
A lot of herbs have been used as brain boosters since ancient times and showed the identical therapeutic effectiveness as contemporary drugs. Healing extracts are derived from their leaves, roots, flowers, or seeds and able to protect our brain from mental diseases.
The following herbs are considered the best brain remedies:
- ginkgo biloba (This plant improves brain qualities, reduces dementia, develops social behavior, and decreases the amount of stress hormones.);
- ginseng (Acting as a potent adaptogen, it promotes both physical and mental energy.);
- lion’s mane (This plant helps to promote concentration and focus as well as reduce depression symptoms.);
- mucuna pruriens (It increases general brain health and acts as a powerful antioxidant.);
- bacopa monnieri (This herb is the best at amplifying memory and learning abilities, acting as a potent nerve and mental tonic.);
- rhodiola rosea (This flower heals brain fog and gives more energy.);
- periwinkle (This plant is able to decrease brain inflammation, to amplify oxygen and glucose circulation, and to help headaches.);
- peppermint (This popular gastronomic plant stimulates creativity, gives energy, and includes a bunch of important minerals.);
- green tea (As a potent antioxidant, it protects the brain from age decline and increases the production of brain cells.);
- Chinese moss (Huperzine A derived from this plant is known for improving memory, treating vascular dementia, and increasing blood circulation.);
- curcumin (This spice amplifies blood flow in the brain and affects new brain cell formation.);
- rosemary (As a strong antioxidant, this sweet herb prevents brain cell death and cures brain inflammation.);
- gotu kola (This plant is good at oxygenating the brain and improving memory functions.);
- ashwagandha (This herb improves task performance and reaction time.);
- sage (It is used as a memory improvement plant, which protects from Alzheimer’s.).
Minerals and vitamins are also crucial construction materials for proper brain structure and functioning. A healthy brainwork is impossible without wholesome nutrients, which prevent it from harmful substances, toxins, stress, and aging factors. Involve into your daily diet magnesium, omega-3 fatty acids, folate, calcium, and vitamin B complex. Their coordinated work helps to cope with panic attacks, anxiety, and mental distress. They postpone brain aging, amplify stress resistance, improve sleep patterns, and increase our mood. Nourish your brain with healthy food and it will repay with gratitude.
Alternative Smart Drugs
“Smart drugs” are considered a new generation of nootropic pills, which became very popular due to abilities to increase cognitive functions. People who suffer from concentration or attention loss, or decreased memory and mental energy can select a proper nootropic and eliminate all disturbing symptoms by a single tablet intake.
The latest and most effective “smart drugs” are offered in the online pharmacy ModafinilXL. This internet store is a proven source that sells qualitative generic nootropics. Modalert, Modvigil, Waklert, Modafresh, Modaheal, Vilafinil, and other modafinil-containing medicines are at your disposal for perfecting your brain functions. All of them improve cognitive abilities in their individual way and can be used without any fear of getting addicted or acquiring adverse reactions.
Numerous human trials prove their effectiveness and safety, that what is acknowledged by our regular customers. These things are really worth trying. Taken in case of need, they make miracles with our apathy, sleepiness, low mood, and fatigue.
Where to Buy Phenibut Safety?
Although Phenibut is not approved in most countries, it can be purchased as a supplement and is available at numerous e-commerce sites and online shops over-the-counter. It is sold as a sleep aid, mood enhancer, and smart drug.
Before buying any brain supplement, think about the possible risks of obtaining side effects, and whether the results are worth getting unpleasant symptoms. It is a very important issue, so do not neglect it. Discuss with a qualified specialist all the advantages and drawbacks of taking Phenibut in your particular case.